反应条件
1: 43 percent / various solvent(s) / 4.5 h / 186 - 190 °C 2: 1) NaH / 1) DMF, 0 deg C, 25 min, 2) DMF, RT, 2 h 3: H2 / 5percent Pd/c / ethanol View Scheme
参考文献
Roth; Tidwell; Ferone; Baccanari; Sigel; DeAngelis; Elwell
Journal of Medicinal Chemistry, 1989 , vol. 32, # 8 p. 1949 - 1958