2-(2,4-二氟苯基)烟酸乙酯合成路线 (共 1 条)
反应条件
sodium carbonate; tetrakis(triphenylphosphine) palladium(0) in ethanol; toluene T=82°C; Inert atmosphere; Product distribution / selectivity;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED; HURREY, Michael; ALARGOV, Dimitar; JOHNSTON, Steven, C.; ROEPER, Stefanie; SNOONIAN, John, R.; COWANS, Brett, A.; VLAHOVA, Petinka; EBERLIN, Alexander; EDDLESTON, Mark; FRAMPTON, Chris
Patent: WO2010/93889 A2, 2010 ;
Location in patent: Page/Page column 45 ;