Stage #1: With palladium 10 on activated carbon; hydrogen in methanol T=20°C; P=2068.65 Torr; Large scale reaction; Stage #2: With hydrogenchloride in methanol T=60 - 65°C; 2 h;
参考文献
Chen, Jian; Przyuski, Katrin; Roemmele, Renee; Bakale, Roger P. Organic Process Research and Development, 2011 , vol. 15, # 5 p. 1063 - 1072