3-甲基-2-[2'-(甲基磺酰基)联苯-4-基]-5-(三氟甲基)喹喔啉合成路线 (共 1 条)
反应条件
potassium phosphate; tetrakis(triphenylphosphine) palladium(0) in 1,4-dioxane T=80°C; Suzuki coupling; 1 h;
参考文献
Hu, Baihua; Unwalla, Rayomand J.; Goljer, Igor; Jetter, James W.; Quinet, Elaine M.; Berrodin, Thomas J.; Basso, Michael D.; Feingold, Irene B.; Nilsson, Annika Goos; Wilhelmsson, Anna; Evans, Mark J.; Wrobel, Jay E.
Journal of Medicinal Chemistry, 2010 , vol. 53, # 8 p. 3296 - 3304