反应条件
1: 100 percent / H2 / 10percent Pd/C / methanol / 1 h 2: 1-hydroxybenzotriazole, N-methylmorpholine, 1-ethyl-3-<(dimethylamino)propyl>carbodiimide hydrochloride / dimethylformamide / 1.) -23 deg C, 2 h, 2.) RT, 16 h View Scheme
参考文献
Rosenberg, Saul H.; Woods, Keith W.; Sham, Hing L.; Kleinert, Hollis D.; Martin, Donald L.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 7 p. 1962 - 1969
