反应条件
1: 2.10 g / p-toluenesulfonic acid / acetone / 1 h / Ambient temperature 2: NH3, HCl / methanol / 0.08 h / Heating 3: NaBH4 / methanol; tetrahydrofuran / 0.5 h 4: aq. sodium periodate / tetrahydrofuran / 24 h / Ambient temperature View Scheme
参考文献
Prugh; Hartman; Mallorga; McKeever; Michelson; Murcko; Schwam; Smith; Sondey; Springer; Sugrue
Journal of Medicinal Chemistry, 1991 , vol. 34, # 6 p. 1805 - 1818
