反应条件
Multi-step reaction with 3 steps 1: 85 percent / pyridine / 24 h / 0 °C2: 75 percent / H2 / 10percent Pd/C / ethanol / 2 h / 1292.9 Torr3: 75 percent / 2,4-bis(4-methoxyphenyl)-1,3-dithia-2,4-diphosphetane 2,4-disulfide / toluene / 12 h / 80 °C
参考文献
Palomino; Meltsner; Kessel; Horwitz Journal of Medicinal Chemistry, 1990 , vol. 33, # 1 p. 258 - 263