反应条件
in tetrahydrofuran; hexane 1.) -78 deg C, 4 h, 2.) from -78 deg C to rt, overnight; Yield given;
参考文献
Williams, Peter D.; Perlow, Debra S.; Payne, Linda S.; Holloway, M. Katharine; Siegl, Peter K. S.; et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 3 p. 887 - 900