反应条件
1: 3,4-dihydro-2H-pyrido[4,3-b]indol-1(5H)-one With sodium hexamethyldisilazane in N,N-dimethyl-formamide T=5°C; 0.333333 h; Inert atmosphere; 2: methyl iodide in N,N-dimethyl-formamide T=5°C; 0.333333 h;
参考文献
AUSPEX PHARMACEUTICALS, INC.
Patent: US2010/113478 A1, 2010 ;
Location in patent: Page/Page column 12 ;