反应条件
1: 1.) NaH / 1.) DMF, 78 deg C, 2.) 78 deg C, 4 h 2: 37 percent / methanol / 1 h / Ambient temperature View Scheme
参考文献
Saxena, Naveen K.; Coleman, Lisa A.; Drach, John C.; Townsend, Leroy B.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 7 p. 1980 - 1983