反应条件
1: 3-methoxy-4-methylbenzoic acid methyl ester With N-bromosuccinmide; 2,2'-azo-bisisobutyronitrile in tetrachloromethane Bromination; 72 h; Heating; 2: pyrrolidine in tetrahydrofuran T=20°C; Alkylation; 2 h; Further stages.;
参考文献
Sall, Daniel J.; Bailey, Dianna L.; Bastian, Jolie A.; Buben, John A.; Chirgadze, Nickolay Y.; Clemens-Smith, Amy C.; Denney, Michael L.; Fisher, Matthew J.; Giera, Deborah D.; Gifford-Moore, Donetta S.; Harper, Richard W.; Johnson, Lea M.; Klimkowski, Valentine J.; Kohn, Todd J.; Lin, Ho-Shen; McCowan, Jefferson R.; Palkowitz, Alan D.; Richett, Michael E.; Smith, Gerald F.; Snyder, David W.; Takeuchi, Kumiko; Toth, John E.; Zhang, Minsheng
Journal of Medicinal Chemistry, 2000 , vol. 43, # 4 p. 649 - 663
