反应条件
1: acetic acid, hydrochloric acid, H2O / 84 h / Heating
2: 89 percent / acetic anhydride / 4 h / Heating
3: Heating
4: LiAlH4 / diethyl ether / 3 h
View Scheme
参考文献
Badger; Schwartz; Picker; Dorman; Bradley; Cheeseman; DiMartino; Hanna; Mirabelli
Journal of Medicinal Chemistry, 1990 , vol. 33, # 11 p. 2963 - 2970