反应条件
1: N,N-dimethyl-formamide With trichlorophosphate T=0°C; 0.5 h; 2: 8-bromo-imidazo[1,2-a]pyridine T=0 - 20°C; 3: With sodium carbonate in water
参考文献
ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC; GIJSEN, Henricus, Jacobus, Maria; MACDONALD, Gregor, James; BISCHOFF, Francois, Paul; TRESADERN, Gary, John; TRABANCO-SUAREZ, Andres, Avelino; VAN BRANDT, Sven, Franciscus, Anna; BERTHELOT, Didier, Jean-Claude
Patent: WO2010/70008 A1, 2010 ;
Location in patent: Page/Page column 52-53 ;
WO 2010/070008 A1