反应条件
1: 98 percent / triethylsilane, BF3 etherate / CH2Cl2 / 0.5 h / 0 °C
2: 1.) BBr3, 2.) water / 1.) -78 deg C to RT, 6 h, CH2Cl2
View Scheme
参考文献
Batt; Maynard; Petraitis; Shaw; Galbraith; Harris
Journal of Medicinal Chemistry, 1990 , vol. 33, # 1 p. 360 - 370