反应条件
1: N-ethyl-N,N-diisopropylamine / 1,4-dioxane / 50 °C 2: iron; acetic acid / 50 °C 3: sodium hydride / N,N-dimethyl acetamide / 0 °C View Scheme
参考文献
Deng, Xianming; Yang, Qingkai; Kwiatkowski, Nicholas; Sim, Taebo; McDermott, Ultan; Settleman, Jeffrey E.; Lee, Jiing-Dwan; Gray, Nathanael S.
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 3 p. 195 - 200