反应条件
1: 1.) 1-hydroxybenzotriazole hydrate, CDI / 1.) THF, 2.) THF, RT, overnight 2: 1N aq. HCl / 2 h / Heating 3: 68 percent / LiAlH4 / tetrahydrofuran / Heating View Scheme
参考文献
Leschke, Christian; Storm, Ruediger; Breitweg-Lehmann, Evelyn; Exner, Torsten; Nuernberg, Bernd; Schunack, Walter
Journal of Medicinal Chemistry, 1997 , vol. 40, # 19 p. 3130 - 3139