1: 4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-yl-amide methanesulphonic salt With methanesulfonic acid in water
T=15 - 105°C; 1.33333 - 1.66667 h; Industry scale;
2: With sodium hydrogencarbonate in water
T=15 - 25°C;
3: methanesulfonyl chloride in water
T=15 - 25°C; 2.5 - 3.75 h; Product distribution / selectivity;