3-(2,3-二氢-7-羟基-1,4-苯并二恶烷-6-基)-1,3-二氢-2H-吲哚-2-酮合成路线 (共 1 条)
反应条件
caesium carbonate in tetrahydrofuran; N,N-dimethyl-formamide T=0 - 25°C; Industry scale;
参考文献
XENON PHARMACEUTICALS INC.
Patent: US2011/87027 A1, 2011 ;
Location in patent: Page/Page column 13 ;