5-溴-n-(2-甲氧基乙基)-3-吡啶甲胺合成路线 （共 2 条）
反应条件
potassium carbonate in acetonitrile T=80°C; 4 h;
参考文献
WO2010/106016 A1, ;
Page/Page column 123 ;
WO 2010/106016 A1
反应条件
potassium acetate; dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in acetonitrile
T=160°C; 0.25 h; Sealed tubeMicrowave irradiation;
参考文献
GLAXO GROUP LIMITED; ALDER, Catherine Mary; BALDWIN, Ian Robert; BARTON, Nicholas Paul; CAMPBELL, Amanda Jennifer; CHAMPIGNY, Aurelie Cecile; HARLING, John David; MAXWELL, Aoife Caitriona; SIMPSON, Juliet Kay; SMITH, Ian Edward David; TAME, Christopher John; WILSON, Caroline; WOOLVEN, James Michael
Patent: WO2011/110575 A1, 2011 ;
Location in patent: Page/Page column 87-88 ;
WO 2011/110575 A1
