反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=20°C; 18 h;
参考文献
De, Surya K.; Barile, Elisa; Chen, Vida; Stebbins, John L.; Cellitti, Jason F.; MacHleidt, Thomas; Carlson, Coby B.; Yang, Li; Dahl, Russell; Pellecchia, Maurizio
Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 8 p. 2582 - 2588