SR 1078; N-[4-[2,2,2-三氟-1-羟基-1-(三氟甲基)乙基]苯基]-4-(三氟甲基)苯甲酰胺合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in dichloromethane T=20°C; 8 h; Inert atmosphere;
参考文献
GRIFFIN, Patrick R.; ROUSH, William R.; KUMAR, Naresh; NUHANT, Philippe; BURRIS, Thomas; SOLT, Laura
Patent: WO2011/115892 A1, 2011 ;
Location in patent: Page/Page column 5; 87; 88 ;
WO 2011/115892 A1