5-氨基-2,3-二氟苯甲腈合成路线 (共 2 条)
反应条件
iron; acetic acid in acetonitrile T=0 - 20°C;
参考文献
SEPRACOR INC.; BURDI, Douglas; SPEAR, Kerry, L.; HARDY, Larry, Wendell
Patent: WO2010/114971 A1, 2010 ;
Location in patent: Page/Page column 237 ;
反应条件
tert.-butylnitrite; copper(I) bromide in acetonitrile T=0 - 20°C;
参考文献
SEPRACOR INC.; BURDI, Douglas; SPEAR, Kerry, L.; HARDY, Larry, Wendell
Patent: WO2010/114971 A1, 2010 ;
Location in patent: Page/Page column 237 ;