5,5-((1R,1R)-哌嗪-1,4-二基双(1-羟基乙烷-2,1-二基))双(4-甲基异苯并呋喃-1(3H)-酮)合成路线 (共 1 条)
反应条件
in ethanol T=150°C; 1.5 h; Microwave irradiation; Product distribution / selectivity;
参考文献
MERCK SHARP andamp;; DOHME CORP.; PASTERNAK, Alexander; SHAHRIPOUR, Aurash; TANG, Haifeng; TEUMELSAN, Nardos, H.; YANG, Lihu; ZHU, Yuping; WALSH, Shawn, P.
Patent: WO2010/129379 A1, 2010 ;
Location in patent: Page/Page column 105-106 ;
WO 2010/129379 A1