反应条件
1.1: thionyl chloride / methanol / 0 - 20 °C 2.1: N-ethyl-N,N-diisopropylamine / N,N-dimethyl-formamide / 20 - 90 °C 3.1: 3-chloro-benzenecarboperoxoic acid / dichloromethane / 0 °C 3.2: 18 h / 95 °C View Scheme
参考文献
Zhu, Aizhi; Zhan, Weiqiang; Liang, Zhongxing; Yoon, Younghyoun; Yang, Hua; Grossniklaus, Hans E.; Xu, Jianguo; Rojas, Mauricio; Lockwood, Mark; Snyder, James P.; Liotta, Dennis C.; Shim, Hyunsuk
Journal of Medicinal Chemistry, 2010 , vol. 53, # 24 p. 8556 - 8568