triethylamine in N,N-dimethyl-formamide T=20°C; 24 h;
参考文献
Merlani, M. I.; Sladkov, V. I.; Parshin, V. A.; Men'shova, N. I.; Levina, I. I.; Suvorov, N. N.
Pharmaceutical Chemistry Journal, 1989 , vol. 23, # 12 p. 950 - 954
Khimiko-Farmatsevticheskii Zhurnal, 1989 , vol. 23, # 12 p. 1431 - 1435
1: 74 percent / NaHCO3 / dimethylformamide / 3 h / 60 - 65 °C 2: 92 percent / Et3N / dimethylformamide / 24 h / 20 °C View Scheme
参考文献
Merlani, M. I.; Sladkov, V. I.; Parshin, V. A.; Men'shova, N. I.; Levina, I. I.; Suvorov, N. N.
Pharmaceutical Chemistry Journal, 1989 , vol. 23, # 12 p. 950 - 954
Khimiko-Farmatsevticheskii Zhurnal, 1989 , vol. 23, # 12 p. 1431 - 1435