反应条件
1: C7H6O2*C13H16N2O2 With sodium carbonate in dichloromethane; water 2: 4-[Pyridin-4-yl]-Benzoic Acid With 4-methyl-morpholine; O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate in N,N-dimethyl-formamide T=20°C;
参考文献
SANOFI; GAUDIN, Christophe; MORYUSEF, Angèle
Patent: WO2014/33221 A1, 2014 ;
Location in patent: Page/Page column 14 ;