反应条件
1: acetonitrile 2: 1.) Zn/Cu, glacial acetic acid, 2.) NH3(g) in MeOH / 1.) DMF, RT, 30 min View Scheme
参考文献
Aerschot, Arthur Van; Everaert, Dirk; Balzarini, Jan; Augustyns, Koen; Jie, Liu; at al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 6 p. 1833 - 1839