反应条件
1: 2.) NH3 (gas) / 1.) reflux, 2.) EtOH, RT, 4 h 2: 75 percent / BCl3 / CH2Cl2 / 4 h / -78 °C 3: 82 percent / 30percent aq. H2O2, 28percent aq. NH4OH / 0.5 h / Ambient temperature View Scheme
参考文献
Bennett, Sharon M.; Nguyen-Ba, Nghe; Ogilvie, Kelvin K.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 8 p. 2162 - 2173
