1-(5-溴-2-氟苯基)吡咯烷合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in 1-methyl-pyrrolidin-2-one T=120°C; 2 h; Sealed vessel;
参考文献
TREVENTIS CORPORATION; REED, Mark, A.; YADAV, Arun; BANFIELD, Scott, C.; BARDEN, Christopher, J.
Patent: WO2012/119035 A1, 2012 ;
Location in patent: Page/Page column 54-55 ;