反应条件
1.1: ammonium acetate / xylene / 5 h / 130 - 135 °C / Industry scale 2.1: potassium acetate / dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct / 1,4-dioxane / 2 h / Inert atmosphere; Reflux 2.2: pH ~ 8 View Scheme
参考文献
PFIZER LIMITED; MILBANK, Jared Bruce John; TRAN, Thien Duc; WAKENHUT, Florian
Patent: WO2011/154871 A1, 2011 ;
