反应条件
1.1: water; lithium hydroxide hydrate / methanol / 2 h / 20 °C 1.2: pH 5 2.1: N-ethyl-N,N-diisopropylamine; ammonium chloride; HATU / N,N-dimethyl-formamide / 2 h / 20 °C View Scheme
参考文献
Blaquiere, Nicole; Do, Steven; Dudley, Danette; Folkes, Adrian; Heald, Robert; Heffron, Timothy; Jones, Mark; Kolesnikov, Aleksandr; Ndubaku, Chudi; Olivero, Alan G.; Price, Stephen; Staben, Steven; Wang, Lan
Patent: US2011/76292 A1, 2011 ;