(1S)-1,5-脱水-1-C-[3-[[5-(4-氟苯基)-2-噻吩基]甲基]-4-甲基苯基]-D-山梨糖醇 2,3,4,6-四(2,2-二甲基丙酸酯)合成路线 (共 1 条)
反应条件
methanol; sodium methylate T=60°C; 16 h; Product distribution / selectivity;
参考文献
JANSSEN PHARMACEUTICA NV; HOUPIS, Ioannis, Nicolaos; LEMAIRE, Sebastien, Francois, Emmanuel
Patent: WO2012/140120 A1, 2012 ;
Location in patent: Page/Page column 92-93 ;
WO 2012/140120 A1