1: With copper(l) iodide; N-ethyl-N,N-diisopropylamine; triphenylphosphine in tetrahydrofuran Sonogashira coupling; 1 h; 2: With bis(dibenzylideneacetone)-palladium(0) in tetrahydrofuran 12 h;
参考文献
McCalmont, William F.; Patterson, Jaclyn R.; Lindenmuth, Michael A.; Heady, Tiffany N.; Haverstick, Doris M.; Gray, Lloyd S.; Macdonald, Timothy L.
Bioorganic and Medicinal Chemistry, 2005 , vol. 13, # 11 p. 3821 - 3839