1-Boc-5-氨基-2,3-二氢吲哚合成路线 (共 4 条)
反应条件
hydrogen; palladium 10 on activated carbon in methanol T=20°C; 1.5 h;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Patent: WO2008/113760 A2, 2008 ;
Location in patent: Page/Page column 92 ;
WO 2008/113760 A2
反应条件
hydrogen; palladium 10 on activated carbon in methanol T=20°C; 1.5 h;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Patent: WO2009/16119 A1, 2009 ;
Location in patent: Page/Page column 54 ;
WO 2009/016119 A1
反应条件
1: 4-(N,N-dimethlyamino)pyridine / tetrahydrofuran / 3 h / 20 - 60 °C 2: hydrogen / palladium 10 on activated carbon / ethanol / 12 h / 20 °C View Scheme
反应条件
1: 4-(N,N-dimethlyamino)pyridine / tetrahydrofuran / 3 h / 20 - 60 °C 2: hydrogen / palladium 10 on activated carbon / ethanol / 12 h / 20 °C View Scheme