1-Boc-6-硝基吲哚啉合成路线 （共 3 条）
反应条件
pyridine; 4-(N,N-dimethlyamino)pyridine in dichloromethane
参考文献
SCHERING CORPORATION; PHARMACOPEIA DRUG DISCOVERY, INC.
Patent: WO2007/24944 A1, 2007 ;
Location in patent: Page/Page column 33-34 ;
WO 2007/024944 A1
反应条件
triethylamine in dichloromethane T=25°C; 16 h;
参考文献
Carruthers, Nicholas I.; Chai, Wenying; Dax, Scott L.; Jablonowski, Jill A.; Li, Xiaobing; Lovenberg, Timothy W.; Murray, William V.; Rudolph, Dale A.; Seierstad, Mark; Youngman, Mark A.
Patent: US2005/70534 A1, 2005 ;
Location in patent: Page/Page column 11 ;
US 20050070534 A1
反应条件
hydrogen; palladium 10 on activated carbon in methanol; ethyl acetate P=760.051 Torr;
参考文献
Carruthers, Nicholas I.; Chai, Wenying; Dax, Scott L.; Jablonowski, Jill A.; Li, Xiaobing; Lovenberg, Timothy W.; Murray, William V.; Rudolph, Dale A.; Seierstad, Mark; Youngman, Mark A.
Patent: US2005/70534 A1, 2005 ;
Location in patent: Page/Page column 11 ;
US 20050070534 A1
