反应条件
sodium hydride 1.) MeCN, RT, 30 min, 2.) a) 0-5 deg C, 15 min, b) RT, overnight; Yield given. Multistep reaction;
参考文献
JANSSEN RandD IRELAND; MC GOWAN, David Craig; LAST, Stefaan Julien; PIETERS, Serge Maria Aloysius; EMBRECHTS, Werner; JONCKERS, Tim Hugo Maria; RABOISSON, Pierre Jean-Marie Bernard
Patent: WO2014/56953 A1, 2014 ;
Location in patent: Page/Page column 8 ;