反应条件
1: 1.) NaH / 1.) MeCN, RT, 30 min, 2.) a) 0-5 deg C, 15 min, b) RT, overnight 2: 88 percent / NaOH / dioxane / 1 h / Heating View Scheme
参考文献
Girgis, Nabih S.; Michael, Maged A.; Smee, Donald F.; Alaghamandan, Hassan A.; Robins, Roland K.; Cottam, Howard B.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 10 p. 2750 - 2755