反应条件
1: 79 percent / KBH4 / methanol / 1.) 0 deg C, 30 min, 2.) RT, 30 min
2: 4-toluenesulfonic acid / toluene / 4.5 h / Heating
View Scheme
参考文献
Buckle, Derek R.; Arch, Jonathon R. S.; Fenwick, Ashley E.; Houge-Frydrych, Catherine S. V.; Pinto, Ivan L.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 11 p. 3028 - 3034
