1: With lithium diisopropyl amide in tetrahydrofuran; n-heptane; ethylbenzene T=-78°C; 2 h; 2: With ammonium chloride in tetrahydrofuran; n-heptane; ethylbenzene
参考文献
Xia, Yan; Jin, Yinglan; Kaur, Navneet; Choi, Yongseok; Lee, Kyeong
European Journal of Medicinal Chemistry, 2011 , vol. 46, # 6 p. 2386 - 2396