4-(三氟甲基)苯并[d]噻唑合成路线 (共 1 条)
反应条件
phosphoric acid; hypophosphorous ether; sodium nitrite 1.) water, 0 deg C, 30 min, 2.) RT; Yield given. Multistep reaction;
参考文献
Mylari; Larson; Beyer; Zembrowski; Aldinger; Dee; Siegel; Singleton
Journal of Medicinal Chemistry, 1991 , vol. 34, # 1 p. 108 - 122