反应条件
1: 92 percent / pyridine / 16 h / Ambient temperature 2: 86 percent / H2 / 10percent Pd-C / ethanol / 6 h / 55 °C / 760 Torr 3: 72 percent / AcOH, H2O / tetrahydrofuran / 14 h / Ambient temperature View Scheme
参考文献
Tanaka; Baba; Hayakawa; Sakamaki; Miyasaka; Ubasawa; Takashima; Sekiya; Nitta; Shigeta; Walker; Balzarini; De Clercq
Journal of Medicinal Chemistry, 1991 , vol. 34, # 1 p. 349 - 357