反应条件
1: triphenylphosphine / 1,2-dichloro-benzene / 12 h / 165 °C
2: hydrogenchloride / 1,4-dioxane; water / 1 h / 20 °C
View Scheme
参考文献
Takeuchi, Tomoki; Oishi, Shinya; Watanabe, Toshiaki; Ohno, Hiroaki; Sawada, Jun-Ichi; Matsuno, Kenji; Asai, Akira; Asada, Naoya; Kitaura, Kazuo; Fujii, Nobutaka
Journal of Medicinal Chemistry, 2011 , vol. 54, # 13 p. 4839 - 4846