1: With n-butyllithium; tri-isopropoxy-borane in tetrahydrofuran; hexane
T=-78°C; 3.17 h;
2: With hydrogenchloride; water in tetrahydrofuran; hexane
T=-78 - 20°C;
参考文献
Cross, R. Matthew; Maignan, Jordany R.; Mutka, Tina S.; Luong, Lisa; Sargent, Justin; Kyle, Dennis E.; Manetsch, Roman
Journal of Medicinal Chemistry, 2011 , vol. 54, # 13 p. 4399 - 4426
