1.1: 4-(N,N-dimethlyamino)pyridine; camphor-10-sulfonic acid; dicyclohexyl-carbodiimide / dichloromethane / 3 h / 20 °C / Inert atmosphere 2.1: methanol; pyridinium p-toluenesulfonate / 6 h / 20 °C / Inert atmosphere 3.1: 4-(N,N-dimethlyamino)pyridine; camphor-10-sulfonic acid; dicyclohexyl-carbodiimide / dichloromethane / 12 h / 20 °C / Inert atmosphere 4.1: methanol; pyridinium p-toluenesulfonate / 24 h / 20 °C / Inert atmosphere 5.1: morpholine; tetrakis(triphenylphosphine) palladium(0) / tetrahydrofuran / 12 h / 20 °C / Inert atmosphere 5.2: Inert atmosphere 6.1: 2,4,6-trichlorobenzoyl chloride; triethylamine / toluene / 1 h / 20 °C / Inert atmosphere 6.2: 7 h / 80 °C 7.1: trifluoroacetic acid / dichloromethane / 5 h / 20 °C / Inert atmosphere View Scheme