1-(4-氨基苯基)-1H-吡啶-2-酮合成路线 (共 2 条)
反应条件
water; ammonium chloride; zinc in tetrahydrofuran; methanol T=20°C;
参考文献
FOREST LABORATORIES HOLDINGS LIMITED
Patent: US2009/239848 A1, 2009 ;
Location in patent: Page/Page column 31 ;
US 20090239848 A1
反应条件
8-hydroxy-quinoline; potassium carbonate; copper(l) iodide in dimethyl sulfoxide T=130°C;
参考文献
WO2006/55951 A2, ;
Page/Page column 59 ;
WO 2006/055951 A2