反应条件
1: N,N-di-isopropylethylamine / N,N-dimethyl-acetamide / 24 h / 100 °C
2: 0.65 g / aq. formic acid / 3 h / Ambient temperature
3: hydrogen / palladium on carbon / ethanol; acetic acid; H2O / 2 h
View Scheme
参考文献
Buck, Ildiko M.; Reese, Colin B.
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1990 , # 11 p. 2937 - 2942