反应条件
trichlorophosphate in N,N-dimethyl-formamide; toluene 1.) RT, 10 min, 2.) reflux, 30 min;
参考文献
Galen, Philip J. M. van; Nissen, Peter; Wijngaarden, Ineke van; IJzerman, Adriaan P.; Soudijn, Willem
Journal of Medicinal Chemistry, 1991 , vol. 34, # 3 p. 1202 - 1206