反应条件
1: NaN3 / ethanol / 3 h / Heating 2: 1.) NaOCH3 / 1.) EtOH, reflux, 20 min, 2.) EtOH, reflux View Scheme
参考文献
Bochis; Chabala; Harris; Peterson; Barash; Beattie; Brown; Graham; Waksmunski; Tischler; Joshua; Smith; Colwell; Wyvratt Jr.; Fisher; Tamas; Nicolich; Schleim; Wilks et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 9 p. 2843 - 2852