反应条件
1: 51 percent / K2CO3, 18-crown-6 / dimethylformamide / 21 h / 110 °C 2: 1.) NaOMe, 2.) 3N HCl / 1.) MeOH, 40 deg C, 2 h, 2.) 50 deg C, 2 h View Scheme
参考文献
Bisacchi; Braitman; Cianci; Clark; Field; Hagen; Hockstein; Malley; Mitt; Slusarchyk; Sundeen; Terry; Tuomari; Weaver; Young; Zahler
Journal of Medicinal Chemistry, 1991 , vol. 34, # 4 p. 1415 - 1421