反应条件
1: potassium phosphate / copper(l) iodide; N-methyl-glycine / N,N-dimethyl-formamide / Reflux 2: AlCl3, aluminium chloride / dichloromethane / 0 - 10 °C 3: sodium hydroxide / tetrahydrofuran / 3 h / 20 °C View Scheme
参考文献
MAPI PHARMA HOLDINGS (CYPRUS) LIMITED; MAROM, Ehud; MIZHIRITSKII, Michael; RUBNOV, Shai
Patent: WO2011/99010 A1, 2011 ;